CAS NO. |
Products Name |
1493694-70-4 |
UNC2250 |
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UNC2250 is a potent and selective Mer inhibitor with IC50 of 1.7 nM, about 160- and 60-fold selectivity over the closely related kinases Axl/Tyro3. |
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418805-02-4 |
PYR41 |
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PYR41 is the first cell-permeable inhibitor of ubiquitin-activating enzyme E1, with no activity at E2. |
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1395084-25-9 |
MS436 |
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MS436 is a diazobenzene-based small-molecule inhibitor for the BRD4 bromodomains with a Ki value of 30-50 nM. |
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218156-96-8 |
SRPIN 340 |
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SRPIN 340 is a selective SRPK inhibitor with Ki of 0.89 μM for SRPK1, showing no significant inhibitory activity against more than 140 other kinases.. |
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725247-18-7 |
XCT790 |
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XCT-790 is a potent, selective and inverse agonist of estrogen-related receptor alpha(ERRα); induces cell death in chemotherapeutic resistant cancer cells. |
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1243583-85-8 |
MG149 |
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MG149 is a selective and potent Tip60 inhibitor with IC50 of 74 uM, similar potentcy for MOF(IC50= 47 uM); little potent for PCAF and p300(IC50 >200 uM). |
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865362-74-9 |
FR 180204 |
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FR180204 is a potent and selective ATP-competitive inhibitor of ERK1 and ERK2 with Ki value of 0.31 uM and 0.14 uM respectively; has IC50 values of 0.51 and 0.33 μM in enzymatic assays against ERK1 and ERK2, respectively. |
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