CAS NO. |
Products Name |
354812-17-2 |
SC-514 |
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SC-514 (GK 01140), a small molecule, is a selective inhibitor of IKK-2; does not inhibit other IKK isoforms or other serine-threonine and tyrosine kinases. |
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202463-68-1 |
AM281 |
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Potent, selective CB1 cannabinoid receptor antagonist/inverse agonist (Ki values are 12 and 4200 nM for CB1 and CB2 receptors respectively). |
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154992-24-2 |
RU-58841 |
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RU 58841 is a specific androgen receptor antagonist or anti-androgen; RU 58841 has a dramatic effect on hair regrowth. |
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104987-11-3 |
Tacrolimus (FK506) |
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FK-506 is a 23-membered macrolide lactone, it reduces peptidyl-prolyl isomerase activity by binding to the immunophilin FKBP12 (FK506 binding protein) creating a new complex. |
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436133-68-5 |
KOBE0065 |
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Kobe0065 is a novel and effective small-molecule compound inhibiting Ras–Raf interaction by SBDD; exhibits potent activity to competitively inhibit the binding of H-Ras·GTP to c-Raf-1 RBD with a Ki value of 46 ± 13 μM. |
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837422-57-8 |
WH-4-023 |
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WH-4-023 is a potent and selective dual Lck/Src inhibitor with IC50 of 2 nM/6 nM for Lck and Src kinase respectively. |
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372196-77-5 |
PIK-75 |
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PIK-75 is a p110α inhibitor with IC50 of 5.8 nM (200-fold more potently than p110β), isoform-specific mutants at Ser773, and also potently inhibits DNA-PK with IC50 of 2 nM. IC50 value: 5.8/2 nM(p110α/DNA-PK) [1] [2] |
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