| CAS NO. |
Products Name |
| 142273-20-9 |
Kenpaullone |
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| Kenpaullone is an ATP-competitive inhibitor of several CDKs (cyclin-dependent kinases) as well as GSK-3β (glycogen synthase kinase 3β). |
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| 1282512-48-4 |
GDC-0032 |
more... |
| GDC-0032 is a potent, next-generation β isoform-sparing PI3K inhibitor targeting PI3Kα/δ/γ with Ki of 0.29 nM/0.12 nM/0.97nM, >10 fold selective over PI3Kβ. |
|
| 667463-85-6 |
BIO-acetoxime |
more... |
| BIO-acetoxime is a potent dual GSK3α/β inhibitor with IC50 of 10 nM, >240-fold selectivity over CDK5/p25, CDK2/cyclin A and CDK1/cyclin B. |
|
| 264218-23-7 |
SB415286 |
more... |
| SB 415286 is a potent and selective cell-permeable, ATP-competitive inhibitor of GSK3α with an IC50 value of 78 nM (similar potency for GSK3β) and a Ki value of 31 nM. |
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| 1047634-65-0 |
GSK2141795 |
more... |
| GSK2141795 is a potent and selective pan-Akt inhibitor with IC50 values of 180 nM for Akt1, 328 nM for Akt2, and 38 nM for Akt3 respectively (Clinical phase 1). |
|
| 305834-79-1 |
sc79 |
more... |
| SC79 is a unique specific Akt activator that may be used to enhance Akt activity in various physiological and pathological conditions. |
|
| 280744-09-4 |
SB216763 |
more... |
| SB 216763 is potent and selective glycogen synthase kinase-3 (GSK-3) inhibitor (Ki = 9 nM); competes with ATP. |
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| 1129669-05-1 |
IM-12 |
more... |
| IM-12 is a potent GSK-3β inhibitor with IC50 of 53 nM; shows a significant activity in several biological tests which was comparable or even outplayed the effects of the known SB-216763. |
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