| CAS NO. |
Products Name |
|
|
| 860352-01-8 |
AZD7762 |
more... |
| AZD7762 is a potent and selective inhibitor of Chk1 with IC50 of 5 nM. It is equally potent against Chk2 and less potent against CAM, Yes, Fyn, Lyn, Hck and Lck. Phase 1 |
|
| 658084-64-1 |
FK866 |
more... |
| APO866 effectively inhibits nicotinamide phosphoribosyltransferase (NMPRTase) with IC50 of 0.09 nM. Phase 1/2 |
|
| 841205-47-8 |
MK-2866 (GTx-024) |
more... |
| MK-2866 (GTx-024) is a selective androgen receptor modulator (SARM) with Ki of 3.8 nM, and is tissue-selective for anabolic organs. Phase 3 |
|
| 401900-40-1 |
Andarine |
more... |
| Andarine is a selective non-steroidal androgen receptor (AR) agonist with Ki of 4 nM, tissue-selective for anabolic organs |
|
| 162831-31-4 |
IEM1754 |
more... |
| IEM 1754 dihydrobroMide is a selective AMPA/kainate receptor blockers for GluR1 and GluR3 with IC50 of 6 μM |
|
| 1240299-33-5 |
AZD3514 |
more... |
| AZD3514 is a potent and oral androgen receptor downregulator with Ki of 2.2 μM and has ability of reducing AR protein expression |
|
| 856925-71-8 |
(-)-Blebbistatin |
more... |
| (-)-Blebbistatin is a cell-permeable inhibitor for non muscle myosin II ATPase with IC50 of ~2 μM, does not inhibit myosin light chain kinase, inhibits contraction of the cleavage furrow without disrupting mitosis or contractile ring assembly |
|
| 1009119-64-5 |
Daclatasvir (BMS790052） |
more... |
| BMS-790052 is a highly selective inhibitor of HCV NS5A with EC50 of 9-50 pM, for a broad range of HCV replicon genotypes and the JFH-1 genotype 2a infectious virus in cell culture. Phase 3 |
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|
|
|
| 659730-32-2 |
AMG517 |
more... |
| AMG 517 is a potent and selective TRPV1 antagonist, antagonizes capsaicin, proton, and heat activation of TRPV1 with IC50 of 0.76 nM, 0.62 nM and 1.3 nM |
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