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Home  All Products |
| All Products >>HER2 // FLT3 |
| CAS NO. |
Products Name |
| 714971-09-2 |
AC480 (BMS-599626) |
more... |
| AC480 (BMS-599626) is a selective and efficacious inhibitor of HER1 and HER2 with IC50 of 20 nM and 30 nM, ~8-fold less potent to HER4, >100-fold to VEGFR2, c-Kit, Lck, MET etc. |
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| 1000669-72-6 |
KW2449 |
more... |
| KW-2449 is a multiple-targeted inhibitor, mostly for Flt3 with IC50 of 6.6 nM, modestly potent to FGFR1, Bcr-Abl and Aurora A; little effect on PDGFRβ, IGF-1R, EGFR. |
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| 301305-73-7 |
TCS359 |
more... |
| TCS 359, a 2-acylaminothiophene-3-carboxamide, is a potent inhibitor of FLT3 with IC50 of 42 nM. |
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| 1327167-19-0 |
BPR1J-097 |
more... |
| BPR1J-097 is a novel small molecule FLT-3 inhibitor(IC50=11±7 nM) with promising in vivo anti-tumour activities; inhibits FLT-3 D835Y with an IC50 of 3 nM. |
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| 923562-23-6 |
FLT3-IN-2 |
more... |
| FLT3-IN-2 is a FLT3 inhibitor with IC50 of ＜ 1 μM, detailed information refer to WO 2012158957 A2 and WO 2007013896. |
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