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Home  All Products |
| All Products >>ATM // ATR |
| CAS NO. |
Products Name |
| 1268524-70-4 |
（+）-JQ1 |
more... |
| (+)-JQ1 is a BET bromodomain inhibitor, with IC50 of 77 nM/33 nM for BRD4(1/2), binding to all bromodomains of the BET family, but not to bromodomains outside the BET family |
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| 1374828-69-9 |
GNE-0877 |
more... |
| GNE0877 is a highly potent, selective, and brain-penetrant aminopyrazole leucine-rich repeat kinase 2 (LRRK2) small molecule inhibitor with an IC50 of 3 nM. |
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| 1232410-49-9 |
VE-821 |
more... |
| VE-821 is a potent and selective ATP competitive inhibitor of ATR with Ki/IC50 of 13 nM/26 nM, shows inhibition of H2AX phosphorylation, minimal activity against PIKKs ATM, DNA-PK, mTOR and PI3Kγ. |
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| 1352226-88-0 |
AZD6738 |
more... |
| AZD6738 is a potent inhibitor of ATR kinase activity with an IC50 of 1 nM against the isolated enzyme and 74 nM against ATR kinase-dependent CHK1 phosphorylation in cells. |
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