CAS NO. |
Products Name |
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792173-99-0 |
SB334867 |
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SB-334867 free base is a selective non-peptide orexin OX1 receptor antagonist with a pKb value of 7.2. |
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1374828-69-9 |
GNE-0877 |
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GNE-0877 is a highly potent and selective leucine-rich repeat kinase 2 (LRRK2) inhibitor with Ki of 0.7 nM. |
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380917-97-5 |
Perampanel |
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Perampanel is a selective noncompetitive AMPA-type glutamate receptor antagonist which has demonstrated anticonvulsant activity in experimental seizure models and antiepileptic activity in clinical trials. |
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441798-33-0 |
Macitentan |
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Macitentan is an orally active, non-peptide, dual ETA/ETB (endothelin) receptor antagonist with IC50 of 0.5 nM/391 nM |
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1219168-18-9 |
BML-275(Dorsomorphin 2HCL) |
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Dorsomorphin is a potent, reversible, selective AMPK inhibitor with Ki of 109 nM, exhibiting no significant inhibition of several structurally related kinases including ZAPK, SYK, PKCθ, PKA, and JAK3. Also inhibits BMP type I receptor. |
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