| CAS NO. |
Products Name |
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| 1186426-66-3 |
DBPR108 |
more... |
| DBPR108 is a DPP4 new orally active selective inhibitor, IC50 value of 15nM, DPP8 and DPP9 no inhibition. |
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| 457081-03-7 |
Pyridone 6 |
more... |
| Pyridone 6 are highly active JAK inhibitors of JAK1 (mice), JAK2 and Tyk2 IC50 15 1 nM and nM,1 nM, respectively, Ki of JAK3 is 5 nM, very low affinity to other protein tyrosine kinase. |
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| 690206-97-4 |
ZM 306416 |
more... |
| ZM 306416 is a VEGFR (Flt and KDR) inhibitor for VEGFR1 with IC50 of 0.33 μM, but also found to inhibit EGFR with IC50 of <10 nM |
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| 446859-33-2 |
RepSox |
more... |
| RepSox is a potent and selective inhibitor of the TGFβR-1/ALK5 with IC50 of 23 nM and 4 nM for ATP binding to ALK5 and ALK5 autophosphorylation in cell-free assays, respectively. |
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